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Selective hydrogenation products of C-076 compounds and derivatives thereof 원문보기

IPC분류정보
국가/구분 United States(US) Patent 등록
국제특허분류(IPC7판)
  • A61K-031/70
  • C07H-017/08
출원번호 US-0928111 (1978-07-31)
발명자 / 주소
  • Chabala John C. (Westfield NJ) Fisher Michael H. (Bridgewater NJ)
출원인 / 주소
  • Merck & Co., Inc. (Rahway NJ 02)
인용정보 피인용 횟수 : 109  인용 특허 : 1

초록 ▼

Derivatives of C-076 are described in which the C-076 molecule, as series of macrolides, has a specific unsaturation, at the 22,23-position, catalytically reduced. Further reaction of the reduced C-076 compounds are also possible. The compounds thus produced have profound anthelmintic, insecticidal,

대표청구항 ▼

A compound having the formula: [Figure] wherein R1 is iso-propyl or sec-butyl; R2 is methoxy, hydroxy or loweralkanoyloxy; and R3 is hydrogen; loweralkanoyl; a4′-loweralkanoyl-a4′-(aa4″-loweralkanoyl-4′-(aa

이 특허에 인용된 특허 (1)

  1. Aoki Atsushi (Sapporo JA) Fukuda Rikiya (Sapporo JA) Nakayabu Toshio (Sapporo JA) Ishibashi Keijiro (Tokyo JA) Takeichi Chiyoko (Tokyo JA) Ishida Mitsuo (Tokyo JA), Antibiotic substances.
    상세보기

이 특허를 인용한 특허 (109)

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