[특허]Transdermal delivery of alpha adrenoceptor blocking agents

Transdermal delivery of alpha adrenoceptor blocking agents 원문보기

IPC분류정보
국가/구분	United States(US) Patent 등록
국제특허분류(IPC7판)	A61F-013/00
출원번호	US-0546106 (1995-10-20)
발명자 / 주소	Santus Giancarlo (Milan ITX) Kim Aeri (Taejon KRX) Francoeur Michael L. (Los Altos CA) Bremer Ulrike (Menlo Park CA)
출원인 / 주소	Flora Inc. (Menlo Park CA 02)
인용정보	피인용 횟수 : 19 인용 특허 : 9

초록

The present invention relates to the transdermal administration of alpha-adrenoceptor blocking compounds. The invention provides methods of administering these compounds to a patient in therapeutically effective amounts.

대표청구항 ▼

A transdermal patch for the delivery of a compound wherein said compound is selected from the group consisting of; 2-cyclohexyl-8-{3-[4-(2-methoxyphenyl)-1-piperazinyl]propylcarbamoyl}-3-methyl-4-oxo-4H-1-benzopyran; 8-{3-[4-(2-methoxyphenyl)-1-piperazinyl]propylcarbamoyl}-3-methyl-4-oxo-2-trifluoromethyl-4H-1-benzopyran; 8-{3-[4-(5-chloro-2-methoxyphenyl)-1-piperazinyl]-propylcarbamoyl}-3-methyl-4-oxo-2-phenyl-4H-1-benzopyran; 8-{3-[4-(5-fluoro-2-methoxyphenyl)-1-piperazinyl]propylcarbamoyl}-3-methyl-4-oxo-2-phenyl-4H-1-benzopyran; 2-cyclohexyl-8-{3-[4-(5-chloro-2-methoxyphenyl)-1-piperazinyl]-propylcarbamoyl}-3-methyl-4-oxo-4H-1-benzopyran; 2-(t-butyl)-7-[3-[4-(5-chloro-2-methoxyphenyl)-1-piperazinyl]-propylcarbamoyl]benzofuran; an enantiomer, a diastereomer, an N-oxide, a prodrug, a metabolite, a prodrug of a metabolite, and a pharmaceutically acceptable salt of said compound to the skin of a patient; said patch comprising a) a backing layer; b) a drug depot selected from the group consisting of a liquid reservoir and a monolithic matrix; said depot comprising said compound, and a permeation enhancer composition; and c) means for affixing the patch to the skin of the patient.

이 특허에 인용된 특허 (9)

Regnier Francois (Nancy FRX), Alfuzosine compositions and use.
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Leonardi Amedeo (Milan ITX) Motta Gianni (Barlassina ITX) Riva Carlo (Varese ITX) Testa Rodolfo (Milan ITX), Benzopyran and benzothiopyran derivatives.
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Leonardi Amedeo (Milan ITX) Motta Gianni (Barlassina ITX) Riva Carlo (Varese ITX) Testa Rodolfo (Milan ITX), Bicyclic heterocyclic derivatives having a1-adrenergic and 5HT₁A.
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Leonardi Amedeo (Milan ITX) Motta Gianni (Barlassina ITX) Riva Carlo (Varese ITX) Guarneri Luciano (Garbagnate Milanese ITX), Flavone derivatives.

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Patel Dinesh C. (Murray UT) Chang Yunik (Lakewood NJ), Penetration enhancement with binary system of oleic acid, oleins, and oleyl alcohol with lower alcohols.

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Yoshida Mitsuhiro (Saitama JPX) Fujimori Hiroyuki (Saitama JPX) Asakawa Hidenori (Saitama JPX) Kasai Masayoshi (Gifu JPX) Kayano Masanori (Saitama JPX) Osawa Shigemitsu (Saitama JPX), Pharmaceutical preparation for percutaneous administration containing bunazosin or its salt.

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Bawa Rajan (Fairport NY), Sustained-release formulation containing and amino acid polymer.

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Gale Robert M. (Los Altos CA) Enscore David J. (Sunnyvale CA), Transdermal delivery of highly ionized fat insoluble drugs.

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Gluchowski Charles (Wayne NJ) Forray Carlos C. (Waldwick NJ) Chiu George (Bridgewater NJ) Branchek Theresa A. (Teaneck NJ) Wetzel John M. (Elmwood Park NJ) Hartig Paul R. (Princeton NJ), Use of a1C specific compounds to treat benign prostatic hyperlasia.

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이 특허를 인용한 특허 (19)

Glenn,Gregory M.; Alving,Carl R., Adjuvant for transcutaneous immunization.
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Carrara,Dario; Porto,Gabriel; Rodriguez,Jorge, Composition for transdermal and/or transmucosal administration of active compounds that ensures adequate therapeutic levels.
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Carrara,Dario Norberto R.; Grenier,Arnaud; Besse,Celine; Simes,Stephen M.; Lehman,Leah M., Formulations for transdermal or transmucosal application.
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Lehman, Leah M.; Simes, Stephen M., Method and apparatus for transdermal or transmucosal application of testosterone.
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Lehman, Leah M.; Simes, Stephen M., Methods and apparatus for transdermal or transmucosal application of testosterone.
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Simes, Stephen M.; Lehman, Leah M., Methods of treating hot flashes with formulations for transdermal or transmucosal application.
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Simes, Stephen M.; Lehman, Leah M., Methods of treating hot flashes with formulations for transdermal or transmucosal application.
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Lee,Youn Joong; Choi,Won Tae; Park,Chan Woo; Kim,Byung Hoon, Output buffer circuit.
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Grenier,Arnaud; Carrara,Dario Norberto R.; Besse,Celine, Permeation enhancing compositions for anticholinergic agents.
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Carrara,R. Dario Norberto; Grenier,Arnaud; Besse,Celine, Pharmaceutical compositions of nicotine and methods of use thereof.
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Tavares, Lino; Shevchuk, Ihor; Alfonso, Mark; Marcenyac, Geraldine; Valia, Kirti H., Terazosin transdermal device and methods.
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Glenn, Gregory M.; Alving, Carl R., Transcutaneous immunization without heterologous adjuvant.
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Carrara, Dario Norberto R.; Grenier, Arnaud, Transdermal compositions for anticholinergic agents.
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Carrara, Dario Norberto R.; Grenier, Arnaud, Transdermal compositions for anticholinergic agents.
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Carrara,R. Dario Norberto; Grenier,Arnaud; Besse,Celine, Transdermal pharmaceutical formulation for minimizing skin residues.
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Carrara, Dario Norberto R.; Grenier, Arnaud, Transdermal testosterone formulation for minimizing skin residues.
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Glenn, Gregory M.; Alving, Carl R., Use of penetration enhancers and barrier disruption agents to enhance the transcutaneous immune response.
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Glenn,Gregory M.; Alving,Carl R., Use of penetration enhancers and barrier disruption methods to enhance the immune response of antigen and adjuvant.
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Glenn, Gregory M.; Cassels, Frederick J., Vaccine for transcutaneous immunization.
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IPC	Description
A	생활필수품
A62	인명구조; 소방(사다리 E06C)
A62B	인명구조용의 기구, 장치 또는 방법(특히 의료용에 사용되는 밸브 A61M 39/00; 특히 물에서 쓰이는 인명구조 장치 또는 방법 B63C 9/00; 잠수장비 B63C 11/00; 특히 항공기에 쓰는 것, 예. 낙하산, 투출좌석 B64D; 특히 광산에서 쓰이는 구조장치 E21F 11/00)
A62B-1/08	.. 윈치 또는 풀리에 제동기구가 있는 것

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Transdermal delivery of alpha adrenoceptor blocking agents 원문보기