4-cycloalkyl-5-substituted pyrimidine compounds useful as crop protection agents
원문보기
IPC분류정보
국가/구분
United States(US) Patent
등록
국제특허분류(IPC7판)
C07D-040/306
C07D-040/106
A01N-043/40
A01N-043/54
출원번호
US-0715293
(1996-09-16)
발명자
/ 주소
Felix Raymond A.
Chin Hsiao-Ling M.
Woolard Frank X.
Lee David L.
Kanne David B.
출원인 / 주소
Zeneca Limited, GB2
대리인 / 주소
Snyder
인용정보
피인용 횟수 :
6인용 특허 :
0
초록▼
Herbicidal 4-cycloalkyl-5-substituted pyrimidine compounds of the formula [ STR 1 ] are described. Herbicidal compositions containing such substituted-pyrimidinyl compounds and methods of controlling undesirable vegetation employing these compounds are also disclosed. The compounds in which XR, is h
Herbicidal 4-cycloalkyl-5-substituted pyrimidine compounds of the formula [ STR 1 ] are described. Herbicidal compositions containing such substituted-pyrimidinyl compounds and methods of controlling undesirable vegetation employing these compounds are also disclosed. The compounds in which XR, is hydroxyl are also useful as intermediates for producing the disclosed substituted-pyrimidinyl derivatives.
대표청구항▼
[ What is claimed is:] [1.] A compound of the formula (I): [ STR 37 ] wherein Z is independently halogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.2 -C.sub.6 alkynyl, nitro, cyano, hydroxy, thiocyano, --N(R.sup.11)(R.sup.12), C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.
[ What is claimed is:] [1.] A compound of the formula (I): [ STR 37 ] wherein Z is independently halogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.6 alkenyl, C.sub.2 -C.sub.6 alkynyl, nitro, cyano, hydroxy, thiocyano, --N(R.sup.11)(R.sup.12), C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 haloalkoxy, (C.sub.1 -C.sub.6)alkoxy-(C.sub.1 -C.sub.6)alkyl, halo(C.sub.1 -C.sub.6)alkoxy-(C.sub.1 -C.sub.6)alkyl, --C(X)--R.sup.10 or --S(O).sub.k --R.sup.10 ;q is 0, 1, 2, 3, 4 or 5;A is C or N;X is oxygen or sulfur;R is hydrogen, hydrocarbyl, hydrocarbyl substituted with one or more of halogen or C.sub.1 -C.sub.6 alkoxy, pyridyl, substituted pyridyl, azabenzyl, pyrimidinyl, substituted pyrimidinyl or is of the formula --C(Y)--R.sup.6, --C(O)--C(O)--R.sup.6, --S(O).sub.2 --R.sup.6, --P(Y)(R.sup.11)(R.sup.12) or --Si(R.sup.13)(R.sup.14)(R.sup.15); reinY is oxygen or sulfur;R.sup.6 is hydrocarbyl, substituted hydrocarbyl, hydrocarbyloxy, substituted hydrocarbyloxy, hydrocarbyl-S--, substituted hydrocarbyl-S--, furyl or is of the formula --N(R.sup.7)(R.sup.8);wherein R.sup.7 and R.sup.8 are each independently hydrogen, hydrocarbyl, substituted hydrocarbyl, hydrocarbyloxy, substituted hydrocarbyloxy, pyridyl, furyl, thienyl, (C.sub.1 -C.sub.6)-alkoxycarbonyl(C.sub.1 -C.sub.6)alkyl, hydroxycarbonyl(C.sub.1 -C.sub.6)alkyl, or N(R.sup.9)(R.sup.10) wherein R.sup.9 and R.sup.10 are each independently hydrogen, C.sub.1 -C.sub.6 alkyl, phenyl or substituted phenyl;or R.sup.7 and R.sup.8 together with the nitrogen to which they are bound form an aziridine, piperazine, morpholine, thiomorpholine, thiomorpholine 1-oxide, thiomorpholine 1-1,dioxide, hexamethyleneimine, piperidine or pyrrolidine ring, any of which may be optionally substituted with C.sub.1 -C.sub.6 alkyl;R.sup.11 and R.sup.12 are each independently C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkylthio or C.sub.1 -C.sub.6 alkoxy;R.sup.13, R.sup.14 and R.sup.15 are each independently C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 haloalkyl, aryl or arylalkyl; andk is 0, 1 or 2;Y.sub.1 is C.sub.3 -C.sub.6 cycloalkyl;Y.sup.2 is independently C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.2 -C.sub.6 alkenyl, C.sub.2 -C.sub.6 alkynyl, mercapto, C.sub.1 -C.sub.6 alkylcarbamylthio, C.sub.1 -C.sub.6 haloalkoxy, nitro, cyano, hydroxy, thiocyano, (C.sub.1 -C.sub.6)-alkoxy-(C.sub.1 -C.sub.6)alkyl, --S(O).sub.k --R.sup.10 or --N(R.sup.11)(R.sup.12), wherein k, R.sup.10, R.sup.11 and R.sup.12 have the same meanings as above; n and m are each independently 0 or 1; and p is 0, 1, or 2; or an agriculturally acceptable salt thereof.
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