Functionalized nitrogen heterocyclic compounds, including benzodiazepines and azasugars, and synthetic methods for preparing such compounds. Nitrogen-containing heterocycles are prepared by reacting amino-carbonyl compounds that contain an amine moiety connected via a linker to a carbonyl moiety wit
Functionalized nitrogen heterocyclic compounds, including benzodiazepines and azasugars, and synthetic methods for preparing such compounds. Nitrogen-containing heterocycles are prepared by reacting amino-carbonyl compounds that contain an amine moiety connected via a linker to a carbonyl moiety with an organoboron derivative.
대표청구항▼
1. A compound of formula wherein:R1 is hydrogen, alkyl, aryl, heteroaryl, hydroxy, or alkoxy; R3 is aryl, heteroaryl, alkenyl, or alkynyl, or R1 and R3 can be joined to form a ring of 5 to 10 atoms; R4 is hydrogen, alkyl, aryl, heteroaryl, alkenyl, alkynyl, acyl, carboxy, or carboxamido. 2. The comp
1. A compound of formula wherein:R1 is hydrogen, alkyl, aryl, heteroaryl, hydroxy, or alkoxy; R3 is aryl, heteroaryl, alkenyl, or alkynyl, or R1 and R3 can be joined to form a ring of 5 to 10 atoms; R4 is hydrogen, alkyl, aryl, heteroaryl, alkenyl, alkynyl, acyl, carboxy, or carboxamido. 2. The compound of claim 1, wherein: the compound has a formula selected from the following: wherein R1 is hydrogen, alkyl, aryl, heteroaryl, hydroxy, or alkoxy; R3 is aryl, heteroaryl, alkenyl or alkynyl; and R4 is hydrogen, alkyl, aryl, heteroaryl, alkenyl, alkynyl, acyl, carboxy, or carboxamido. 3. The compound of claim 1, wherein:R3 is aryl, heteroaryl, or alkenyl, and R4 is hydrogen.
연구과제 타임라인
LOADING...
LOADING...
LOADING...
LOADING...
LOADING...
이 특허에 인용된 특허 (32)
Nicolaou Kyriacos C. (Havertown PA) Petasis Nicos A. (Drexel Hill PA) Li Wen-Sen (Philadelphia PA) Ladduwahetty Tamara (Philadelphia PA) Randall Jared L. (Philadelphia PA) Webber Stephen E. (Philadel, Alkanoarachidonic acids.
Savoca Ann C. L. (Sinking Springs PA) Louie Michael (Bethlehem PA), Amine-boron adducts as reduced odor catalyst compositions for the production of polyurethanes.
Bell Robert T. (Garland TX) Platt Richard B. (Allen TX), Bridging and signalling subsystems and methods for private and hybrid communications systems including multimedia system.
Weinberg W. Henry ; McFarland Eric ; Goldwasser Isy ; Boussie Thomas ; Turner Howard ; Van Beek Johannes A. M. ; Murphy Vince ; Powers Timothy, Combinatorial synthesis and analysis of organometallic compounds and catalysts.
Hughes James P. ; Olson Steve A., Policy caching method and apparatus for use in a communication device based on contents of one data unit in a subset of.
Wong Chi-Huey (Rancho Santa Fe CA) Kajimoto Tetsuya (Kumamoto CA JPX) Liu Kun-Chin (San Diego CA) Chen Lihren (San Diego CA), Process for forming omega-deuxy-azasugars.
Bruce David Alan ; White Mark Gilmore ; Bertrand Joseph Aaron ; Dai Pei-Shing Eugene ; Petty Randall Hughes, Synthesis of metal--containing aluminophosphates with layered structure.
Jeffrey Conklin ; David Foucher ; Daniel Foucher, System and method for representing data and providing electronic non-repudiation in a negotiations system.
Opalka Zbigniew ; Aggarwal Vijay ; Kong Thomas ; Firth Christopher ; Costantino Carl, System architecture for and method of processing packets and/or cells in a common switch.
Deborah L. Caswell ; Srinivas Ramanathan ; James D. Hunter ; Scott S. Neal ; Frederick A. Sieker ; Mark D. Smith, Template-driven approach for generating models on network services.
Harrison, Bryce Alden; Kimball, Spencer David; Mabon, Ross; Rawlins, David Brent; Goodwin, Nicole C, Inhibitors of sodium glucose co-transporter 2 and methods of their use.
Giguere, Joshua Robert; McCarthy, Keith Edward; Reisch, Helge Alfred; Sandoval, Sergio; Stymiest, Jake Larry, Transition metal-catalyzed processes for the preparation of N-allyl compounds and use thereof.
※ AI-Helper는 부적절한 답변을 할 수 있습니다.