최소 단어 이상 선택하여야 합니다.
최대 10 단어까지만 선택 가능합니다.
다음과 같은 기능을 한번의 로그인으로 사용 할 수 있습니다.
NTIS 바로가기Journal of molecular structure, v.1289, 2023년, pp.135780 -
S, Anjali , M, Sangeetha , M, Nithya , Krishnan, Gopika V. , Varughese, Sunil , Kumar, B.S. Dileep , N, Srikantamurthy , D, Shridevi , Somappa, Sasidhar B.
초록이 없습니다.
Appl. Microbiol. Biotechnol. Kardos 92 677 2011 10.1007/s00253-011-3587-6 Penicillin: the medicine with the greatest impact on therapeutic outcomes
Nature Brown 529 336 2016 10.1038/nature17042 Antibacterial drug discovery in the resistance era
Chem. Commun. Galloway 2446 2009 10.1039/b816852k The discovery of antibacterial agents using diversity-oriented synthesis
J. Med. Chem. Sun 65 436 2022 10.1021/acs.jmedchem.1c01592 Natural berberine-derived azolyl ethanols as new structural antibacterial agents against drug-resistant escherichia coli
J. Med. Chem. Dewangan 65 5433 2022 10.1021/acs.jmedchem.1c01809 Spermine-conjugated short proline-rich lipopeptides as broad-spectrum intracellular targeting antibacterial agents
J. Med. Chem. Liang 65 14221 2022 10.1021/acs.jmedchem.2c01437 Design and synthesis of phenyl sulfide-based cationic amphiphiles as membrane-targeting antimicrobial agents against gram-positive pathogens
J. Med. Chem. Legru 65 16392 2022 10.1021/acs.jmedchem.2c01257 Optimization of 1,2,4-triazole-3-thiones toward broad-spectrum metallo-β-lactamase inhibitors showing potent synergistic activity on VIM- and NDM-1-producing clinical isolates
ACS Biol. Med. Chem. Au Alkhzem 2 607 2022 10.1021/acsbiomedchemau.2c00033 Practical synthesis of antimicrobial long linear polyamine succinamides
J. Med. Chem. Mała 65 14180 2022 10.1021/acs.jmedchem.2c01373 Discovery of N‑β‑l‑fucosyl amides as high-affinity ligands for the Pseudomonas aeruginosa Lectin LecB
J. Med. Chem. Verma 65 4085 2022 10.1021/acs.jmedchem.1c01909 Discovery of inhibitors of the lipopolysaccharide transporter msba: from a screening hit to potent wild-type gram-negative activity
J. Med. Chem. Xie 65 6171 2022 10.1021/acs.jmedchem.2c00001 Unique carbazole-oxadiazole derivatives as new potential antibiotics for combating gram-positive and -negative bacteria
Anti Infective Agents Bhat 17 66 2018 10.2174/2211352516666180914101758 Anti-mitotic activity of the benzothiazole-pyrazole hybrid derivatives
Bioorg. Med. Chem. Lett. Ningaiah 23 4532 2013 10.1016/j.bmcl.2013.06.042 Novel pyrazoline amidoxime and their 1,2,4-oxadiazole analogues: Synthesis and pharmacological screening
Eur. J. Med. Chem. Vijesh 62 410 2013 10.1016/j.ejmech.2012.12.057 New pyrazole derivatives containing 1,2,4-triazoles and benzoxazoles as potent antimicrobial and analgesic agents
Biomedicines Ebenezer 10 1 2022 10.3390/biomedicines10051124 A review of the recent development in the synthesis and biological evaluations of pyrazole derivatives
Arch. Pharm. Bekhit 338 167 2005 10.1002/ardp.200400940 Novel pyrazole derivatives as potential promising anti-inflammatory antimicrobial agents
Dye. Pigment. Karci 80 47 2009 10.1016/j.dyepig.2008.05.001 The synthesis, antimicrobial activity and absorption characteristics of some novel heterocyclic disazo dyes
Eur. J. Med. Chem. Dai 166 470 2019 10.1016/j.ejmech.2019.01.070 Excellent antitumor and antimetastatic activities based on novel coumarin/pyrazole oxime hybrids
ChemistrySelect Kuthyala 5 10827 2020 10.1002/slct.202002483 Synthesis, characterization, and anticancer studies of some pyrazole-based hybrid heteroatomics
Bioorg. Med. Chem. Lett. Ranatunge 14 6049 2004 10.1016/j.bmcl.2004.09.073 3-(2-Methoxytetrahydrofuran-2-yl)pyrazoles: a novel class of potent, selective cyclooxygenase-2 (COX-2) inhibitors
J. Med. Chem. Bailey 28 256 1985 10.1021/jm00380a020 3, 4-diphenyl-1H-pyrazole-1-propanamine antidepressants
RSC Adv. Viveka 5 94786 2015 10.1039/C5RA17391D Design, synthesis, anticonvulsant and analgesic studies of new pyrazole analogues: A Knoevenagel reaction approach
Bioorg. Chem. Pogaku 93 2019 10.1016/j.bioorg.2019.103307 Design, synthesis, molecular modelling, ADME prediction and anti-hyperglycemic evaluation of new pyrazole-triazolopyrimidine hybrids as potent α-glucosidase inhibitors
J. Med. Chem. Penning 40 1347 1997 10.1021/jm960803q Synthesis and biological evaluation of the 1,5-diarylpyrazole class of cyclooxygenase-2 inhibitors: Identification of 4-[5-(4-methylphenyl)- 3(trifluoromethyl)-1h-pyrazol-1-yl]benzenesulfonamide (sc-58635, celecoxib)
Br. J. Pharmacol. Hosie 115 909 1995 10.1111/j.1476-5381.1995.tb15896.x Actions of the insecticide fipronil, on dieldrin-sensitive and - resistant GABA receptors of Drosophila melanogaster
Rev. Med. Brux. Wespes 19 437 1998 Sildenafil
Nucleosides Nucleotides Nucleic Acids Elgemeie 38 183 2019 10.1080/15257770.2018.1508693 Novel synthesis and biological evaluation of the first pyrazole thioglycosides as pyrazofurin analogues
Bioorg. Med. Chem. Bekhit 12 1935 2004 10.1016/j.bmc.2004.01.037 Design, synthesis and biological evaluation of some pyrazole derivatives as anti-inflammatory-antimicrobial agents
Org. Commun. Chate 5 83 2012 Synthesis and antimicrobial screening of novel 2-(5-(4-(allyloxy)-3-methoxyphenyl)-1H-pyrazol-3-yl)phenols analogues of 2-(4-(allyloxy)-3-methoxyphenyl)-4H-chromen-4-ones
Bioorg. Med. Chem. Lett. Li 25 5052 2015 10.1016/j.bmcl.2015.10.028 Synthesis and biological evaluation of 1,3-diaryl pyrazole derivatives as potential antibacterial and anti-inflammatory agents
Anal. Chem. Lett. Desai 10 307 2020 10.1080/22297928.2020.1785325 Antimicrobial activity and molecular docking of pyrazole bearing the benzodiazepine moiety
Indian J. Chem. Sect. B Org. Med. Chem. Desai 59 238 2020 Synthesis and antimicrobial activity of some hybrid 2-aryl-4-(1-phenyl-3-(p-tolyl)-1H-pyrazol-4-yl)-2,3-dihydro-1H-benzo[b][1,4]diazepine derivatives
Bioorg. Med. Chem. Bozorov 27 3511 2019 10.1016/j.bmc.2019.07.005 1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: a recent overview
J. Med. Chem. Kumari 63 12290 2020 10.1021/acs.jmedchem.0c00530 Amide bond bioisosteres: strategies, synthesis, and successes
J. Mol. Struct. Gökalp 1212 2020 10.1016/j.molstruc.2020.128140 Triazole based azo molecules as potential antibacterial agents: Synthesis, characterization, DFT, ADME and molecular docking studies
Nucleosides Nucleotides Noble 10 487 1991 10.1080/07328319108046503 Synthesis and biological evaluation of carbocyclic analogues of ribavirin
Henry Ford Hosp. Med. J. Kiani 26 12 1978 In vitro and clinical studies of cefaclor, a new cephalosporin
Anticancer Res. Perabo 24 2869 2004 Carboxyamido-triazole (CAI), a signal transduction inhibitor induces growth inhibition and apoptosis in bladder cancer cells by modulation of Bcl-2
Eur. J. Med. Chem. Hassan 171 332 2019 10.1016/j.ejmech.2019.03.052 New pyrazole derivatives: Synthesis, anti-inflammatory activity, cycloxygenase inhibition assay and evaluation of mPGES
RSC Adv. Singh 4 19013 2014 10.1039/C4RA02649G Design, synthesis and mode of action of some benzothiazole derivatives bearing an amide moiety as antibacterial agents
Res. Pharm. Sci. Egbujor 17 99 2022 10.4103/1735-5362.329930 Design, synthesis, and molecular docking of cysteine-based sulphonamide derivatives as antimicrobial agents
RSC Adv. Zhou 9 41173 2019 10.1039/C9RA09287K Synthesis and biological activities of local anesthetics
10.1128/AAC.14.4.557 I. Vivo, A. Activities, SCE-963, a New Broad-Spectrum Cephalosporin : In Vitro and In Vivo Antibacterial Activities, 14 (1978).
Polyhedron Borrás 19 1859 2000 10.1016/S0277-5387(00)00474-5 Coordination chemistry of sulfamethizole: crystal structures of [Cu(sulfamethizolate)2(py)2(OH2)]·H2O, [M(sulfamethizolate)2(py)2(OH2)2] [M = Co and Ni] and {Cu(sulfamethizolate)2(dmf)2}(∞)
J. Indian Chem. Soc. Elangovan 98 2021 10.1016/j.jics.2021.100144 Synthesis, spectral and quantum mechanical studies and molecular docking studies of Schiff base (E)2-hydroxy-5-(((4-(N-pyrimidin-2-yl)sulfamoyl)phenyl)imino)methyl benzoic acid from 5-formyl salicylic acid and sulfadiazine
Bioorg. Chem. Jalaja 108 2021 10.1016/j.bioorg.2021.104664 Anti-hyperlipidemic potential of natural product based labdane-pyrroles via inhibition of cholesterol and triglycerides synthesis
Bioorg. Chem. Anaga 105 2020 10.1016/j.bioorg.2020.104375 Advanced glycation end-products (AGE) trapping agents: Design and synthesis of nature inspired indeno[2,1-c]pyridinones
ACS Med. Chem. Lett. Jalaja 9 662 2018 10.1021/acsmedchemlett.8b00109 Discovery of natural product derived labdane appended triazoles as potent pancreatic lipase inhibitors
J. Org. Chem. Ashitha 83 113 2018 10.1021/acs.joc.7b02463 BF3·OEt2-mediated tandem annulation: a strategy to construct functionalized chromeno- and pyrano-fused pyridines
Monatshefte Fur Chem. Somappa 146 2067 2015 10.1007/s00706-015-1476-x A one-pot synthesis of indole-appended heterocycles as potent anti-inflammatory, analgesic, and CNS depressant agents
ACS Omega Salfeena 3 8074 2018 10.1021/acsomega.8b01017 Synthesis of 1,2,4-Trisubstituted-(1 H)-imidazoles through Cu(OTf)2-/I2-Catalyzed C-C Bond Cleavage of Chalcones and Benzylamines
Org. Biomol. Chem. Salfeena 14 10165 2016 10.1039/C6OB02133F BF3·Et2O mediated one-step synthesis of N-substituted-1,2-dihydropyridines, indenopyridines and 5,6-dihydroisoquinolines
Chem. Biol. Drug Des. Praveen Kumar 90 703 2017 10.1111/cbdd.12990 Antibacterial and antitubercular evaluation of dihydronaphthalenone-indole hybrid analogs
Med. Chem. Res. Sasidhar 22 3518 2013 10.1007/s00044-012-0370-x Synthesis of some bisindolyl analogs for in vitro cytotoxic and DNA cleavage studies
ChemistrySelect Mohan 3 6394 2018 10.1002/slct.201801126 Functionalized pyrimidines from alkynes and nitriles: application towards the synthesis of marine natural product meridianin analogs
Appl. Organomet. Chem. Kempasiddhaiah 33 1 2019 10.1002/aoc.4846 Magnetite tethered mesoionic carbene-palladium (II): an efficient and reusable nanomagnetic catalyst for Suzuki-Miyaura and Mizoroki-Heck cross-coupling reactions in aqueous medium
Russ. J. Gen. Chem. Basavanna 91 2257 2021 10.1134/S1070363221110128 A new series of 1,3,4-oxadiazole linked quinolinyl-pyrazole/isoxazole derivatives: synthesis and biological activity evaluation
Eur. J. Org. Chem. Silva 4348 2004 10.1002/ejoc.200400407 3(5) -(2-Hydroxyphenyl) -5(3)-styrylpyrazoles synthesis and diels alder transformations
Bioorg. Med. Chem. Lett. Goher 29 449 2019 10.1016/j.bmcl.2018.12.025 Development of novel liver X receptor modulators based on a 1,2,4-triazole scaffold
Org. Lett. Kumar 22 4620 2020 10.1021/acs.orglett.0c01237 Ru(II)-catalyzed oxidative olefination of benzamides: switchable aza-michael and aza-wacker reaction for synthesis of isoindolinones
Bull. Korean Chem. Soc. Farooq 41 918 2020 10.1002/bkcs.12088 Microwave-assisted synthesis and molecular docking study of heteroaromatic chalcone derivatives as potential antibacterial agents
10.26655/JMCHEMSCI.2022.2.11 Gaikwad, M., Gaikwad, S., Kamble, R. Journal of medicinal and chemical sciences synthesis of novel series of 1- (6-Hydroxy-4- (1 H -indol-3-yl) -3, 6- evaluations of their antimicrobial activity with insilco docking study, 5 (2022) 239-248. doi:10.26655/JMCHEMSCI.2022.2.11.
Clinical and Laboratory Standards Institute, Performance Standards for Antimicrobial Disk Susceptibility Tests: Approved Standard - Eleventh edition, 2012. M02-A11.
Int. J. Pharm. Sci. Rev. Res. Bailey-shaw 47 145 2017 In-vitro evaluation of the anti-inflammatory potential of selected Jamaican plant extracts using the Bovine Serum albumin protein denaturation assay
Bioinformation Chandra 10 288 2014 10.6026/97320630010288 Molecular docking studies of benzimidazopyrimidine and coumarin substituted benzimidazopyrimidine derivatives: as potential human Aurora A kinase inhibitors
*원문 PDF 파일 및 링크정보가 존재하지 않을 경우 KISTI DDS 시스템에서 제공하는 원문복사서비스를 사용할 수 있습니다.
※ AI-Helper는 부적절한 답변을 할 수 있습니다.