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NTIS 바로가기Journal of medicinal chemistry, v.55 no.8, 2012년, pp.3687 - 3698
Lee, Won-Gil (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea) , Lee, So-Deok (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea) , Cho, Joong-Heui (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea) , Jung, Younghwan (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea) , Kim, Jeong-hyun (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea) , Hien, Tran T. (College of Pharmacy,Seoul National University, Seoul, Republic of Korea) , Kang, Keon-Wook (College of Pharmacy,Seoul National University, Seoul, Republic of Korea) , Ko, Hyojin (Graduate Program of Medical System Engineering,Gwangju Institute of Science and Technology (GIST), Gwangju 500-712,Republic of Korea) , Kim, Yong-Chul (School of Life Sciences, GwangjuInstitute of Science and Technology (GIST), Gwangju 500-712, Republicof Korea)
Screening of a library of chemical compounds showed that the dichloropyridine-based analogue 9 was a novel P2X(7) receptor antagonist. To optimize its activity, we assessed the structure-activity relationships (SAR) of 9, focusing on the hydrazide linker, the dichloropyridine skeleton, and the hydro...
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