The present invention relates to novel C(29)-oximinomilbemycin derivatives of formula I, to their preparation and to the use thereof for controlling pests. The invention further relates to pesticidal compositions which contain at least one of these compounds as active ingredient. The novel compounds
The present invention relates to novel C(29)-oximinomilbemycin derivatives of formula I, to their preparation and to the use thereof for controlling pests. The invention further relates to pesticidal compositions which contain at least one of these compounds as active ingredient. The novel compounds have the general formula I [Figure] (I) wherein X is a group selected from -CH(OR1)-, -C(O)-or -C(〓N-OR)-, R1 is hydrogen or a OH protective group, R is hydrogen, a OH protective group, an alkyl, cycloalkyl or acyl group, R2 is methyl, ethyl, isopropyl, sec-butyl or the [Figure] wherein A is methyl, ethyl or isopropyl; and R3 is hydrogen, C1-C6alkyl, C2-C6alkenyl, a radial selected from the group consisting of phenyl and benzyl which is unsubstituted or substituted by one or more members selected from the group consisting of halogen, C1-C3alkyl, C1-C3alkoxy, C1-C3alkylthio, C1-C3haloalkyl, nitro or cyano, or is the group U [Figure] (U) wherein n is 0, 1, 2, 3, 4 or 5, E is oxygen or -CH(Rd)-and Rz is hydrogen, Ra is hydrogen, halogen, C1-C3alkyl, C1-C3alkoxy or 2-tetrahydropyranyl, and Rb, Rc and Rd are each independently hydrogen, halogen, C1-C3alkyl or C1-C3alkoxy, which group U may also be in unsaturated form.
대표청구항▼
A compound of formula I [Figure] (I) wherein X is a group selected from -CH(OR1)-, R2 is methyl, ethyl, isopropyl, sec-butyl or the [Figure] wherein A is methyl, ethyl or isopropyl; and R3 is hydrogen, C1-C6alkyl, C2-C6alkenyl, a radial selected from the group consisting of phenyl and benzyl which i
A compound of formula I [Figure] (I) wherein X is a group selected from -CH(OR1)-, R2 is methyl, ethyl, isopropyl, sec-butyl or the [Figure] wherein A is methyl, ethyl or isopropyl; and R3 is hydrogen, C1-C6alkyl, C2-C6alkenyl, a radial selected from the group consisting of phenyl and benzyl which is unsubstituted or substituted by one or more members selected from the group consisting of halogen, C1-C3alkyl, C1-C3alkoxy, C1-C3alkylthio, C1-C3haloalkyl, nitro or cyano, or is the group U [Figure] (U) wherein n is 0, 1, 2, 3, 4 or 5, E is oxygen or -CH(Rd)-and Rz is hydrogen, Ra is hydrogen, halogen, C1-C3alkyl, C1-C3alkoxy or 2-tetrahydropyranyl, and Rb, Rc and Rd are each independently hydrogen, halogen, C1-C3alkyl or C1-C3alkoxy, which group U may also be in unsaturated form.
연구과제 타임라인
LOADING...
LOADING...
LOADING...
LOADING...
LOADING...
이 특허에 인용된 특허 (4)
Chabala John C. (Westfield NJ) Fisher Michael H. (Bridgewater NJ) Mrozik Helmut H. (Matawan NJ), 13-Halo and 13-deoxy derivatives of C-076 compounds.
Soll, Mark David; Cramer, Luiz Gustavo; Pate, James; Shub, Natalya; Le Hir de Fallois, Loic Patrick; Timmons, Philip Reid, Compositions comprising an aryl pyrazole and/or a formamidine, methods and uses thereof.
Soll, Mark David; Cramer, Luiz Gustavo; Wurtz, Patrice; Pate, James; Shub, Natalya; Le Hir de Fallois, Loic Patrick; Timmons, Philip Reid, Compositions comprising an aryl pyrazole and/or a formamidine, methods and uses thereof.
Maulding Donald R. (57 Katydid Dr. Somerville NJ) Kumar Anil (36-C Needham Way Princeton NJ), Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds.
※ AI-Helper는 부적절한 답변을 할 수 있습니다.