초록 ▼

This invention concerns compounds of formula. [EQU1]stereochemically isomeric forms thereof, acid or base addition salts thereof, N-oxides thereof, or quaternary ammonium derivatives thereof, wherein the dotted line is an optional bond; X is a direct bond when the dotted line represents a bond, or X

This invention concerns compounds of formula. [EQU1]stereochemically isomeric forms thereof, acid or base addition salts thereof, N-oxides thereof, or quaternary ammonium derivatives thereof, wherein the dotted line is an optional bond; X is a direct bond when the dotted line represents a bond, or X is hydrogen or hydroxy, when the dotted line does not represent a bond; R1, R2, R5 and R6 are each independently selected from hydrogen, halo, hydroxy, C1-4alkyl, C1-4alkyloxy, -SO3H, and the like; R3 and R4 are each independently selected from hydrogen, halo, hydroxy, C1-4alkyl, C1-4alkyloxy, nitro, amino, cyano, trifluoromethyl, or trifluoromethoxy; L is a radical of formula [EQU2]wherein A1 is a direct bond or C1-6alkanediyl; A2 is C2-6alkanediyl; and R7 to R11 are hydrogen, C1-6alkyl, aminoC1-6alkyl and the like; having biocidal properties; their preparation, compositions containing them and their use as a biocide.

대표청구항 ▼

1. A compound of formula (I) [EQU38]a stereochemically isomeric form thereof, an acid or base addition salt thereof, an N-oxide thereof, or a quaternary ammonium derivative thereof, wherein the dotted line is an optional bond; X is a direct bond when the dotted line represents a bond, or X is hydrog

1. A compound of formula (I) [EQU38]a stereochemically isomeric form thereof, an acid or base addition salt thereof, an N-oxide thereof, or a quaternary ammonium derivative thereof, wherein the dotted line is an optional bond; X is a direct bond when the dotted line represents a bond, or X is hydrogen or hydroxy, when the dotted line does not represent a bond; R1 and R2 are each independently selected from hydrogen, halo, hydroxy, C1-4alkyl, C1-4alkyloxy, nitro, amino, cyano, trifluoromethyl, trifluoromethoxy, C1-6alkylcarbonyl hydroxycarbonyl, C1-6alkyloxycarbonyl, aminocarbonyl, di(C1-4alkyl)aminocarbonyl, C1-6alkylsulfinyl, C1-6alkylsulfonyl, aminosulfonyl, di(C1-4alkyl)aminosulfonyl, or -SO3H; R3 and R4 are each independently selected from hydrogen, halo, hydroxy, C1-4alkyl, C1-4alkyloxy, nitro, amino, cyano, trifluoromethyl, or trifluoromethoxy; R5 and R6 are each independently selected from hydrogen, halo, hydroxy, C1-4alkyl, C1-4alkyloxy, nitro, amino, cyano, trifluoromethyl, trifluoromethoxy, C1-6alkylcarbonyl, hydroxycarbonyl, C1-6alkyloxycarbonyl, aminocarbonyl, di(C1-4alkyl)aminocarbonyl, C1-6alkylsulfinyl, C1-6alkylsulfonyl, aminosulfonyl, di(C1-4alkyl)aminosulfonyl, or -SO3H, L is a radical of formula [EQU39] wherein A1 is a direct bond or C1-6alkanediyl; A2 is C2-6alkanediyl; R7 is hydrogen, C1-4alkyl, phenyl or benzyl; R8 and R9 are each independently hydrogen, C1-6alkyl, aminoC1-6alkyl or mono- or di(C1-4alkyl)aminoC1-6alkyl; R10 is hydrogen, C1-6alkyl, aminoC1-6alkyl or mono- or di(C1-4alkyl)aminoC1-6alkyl; and R11 is hydrogen, C1-6alkyl, amino, aminoC1-6alkyl or mono- or di(C1-4alkyl)aminoC1-6alkyl; provided that when L is a radical of formula (a-9) then R11 is other than hydrogen.