$\require{mediawiki-texvc}$

연합인증

연합인증 가입 기관의 연구자들은 소속기관의 인증정보(ID와 암호)를 이용해 다른 대학, 연구기관, 서비스 공급자의 다양한 온라인 자원과 연구 데이터를 이용할 수 있습니다.

이는 여행자가 자국에서 발행 받은 여권으로 세계 각국을 자유롭게 여행할 수 있는 것과 같습니다.

연합인증으로 이용이 가능한 서비스는 NTIS, DataON, Edison, Kafe, Webinar 등이 있습니다.

한번의 인증절차만으로 연합인증 가입 서비스에 추가 로그인 없이 이용이 가능합니다.

다만, 연합인증을 위해서는 최초 1회만 인증 절차가 필요합니다. (회원이 아닐 경우 회원 가입이 필요합니다.)

연합인증 절차는 다음과 같습니다.

최초이용시에는
ScienceON에 로그인 → 연합인증 서비스 접속 → 로그인 (본인 확인 또는 회원가입) → 서비스 이용

그 이후에는
ScienceON 로그인 → 연합인증 서비스 접속 → 서비스 이용

연합인증을 활용하시면 KISTI가 제공하는 다양한 서비스를 편리하게 이용하실 수 있습니다.

Methods for synthesis of acyloxyalkyl derivatives of GABA analogs 원문보기

IPC분류정보
국가/구분 United States(US) Patent 등록
국제특허분류(IPC7판)
  • C07C-271/22
  • C07C-271/00
출원번호 US-0460091 (2003-06-11)
발명자 / 주소
  • Raillard,Stephen P.
  • Zhou,Cindy X.
  • Yao,Fenmei
  • Manthati,Suresh Kumar
  • Xiang,Jia Ning
  • Gallop,Mark A.
출원인 / 주소
  • Xenoport, Inc.
대리인 / 주소
    Dorsey & Whitney LLP
인용정보 피인용 횟수 : 23  인용 특허 : 55

초록

초록이 없습니다.

대표청구항

대표청구항이 없습니다.

이 특허에 인용된 특허 (55)

  1. Alexander Jose (Lawrence KS), (Acyloxyalkoxy)carbonyl derivatives as bioreversible prodrug moieties for primary and secondary amine functions in drugs.
    상세보기
  2. Lin Yang-I (Tappan NY) Bitha Panayota (Nanuet NY) Sakya Subas (Pomona NY) Strohmeyer Timothy W. (Demarest NJ) Bush Karen (Princeton NJ) Ziegler Carl B. (Pearl River NY) Feigelson Gregg B. (Airmont NY, 2-thiosubstituted carbapenems.
    상세보기
  3. Alexander Jose (Lawrence KS), Acyloxyisopropyl carbamates as prodrugs for amine drugs.
    상세보기
  4. Saunders Richard J. (San Jose CA) Mefferd Wayne Sherman (Los Altos Hills CA), Apparatus for tracking moving workpiece by a laser beam.
    상세보기
  5. Lund Frantz J. (Lyngby DKX), Aryloxymethylcarbonochloridate ester intermediates for use in synthesizing pro drugs and their use therefor.
    상세보기
  6. Guindon Yvan (Closse Ile Bizard CAX) Girard Yves (Pierrefonds CAX) Lau Cheuk K. (Pierrefonds CAX) Fortin Rejean (Montreal CAX) Rokach Joshua (Laval CAX) Yoakim Christiane (Montreal CAX), Benzo[A]phenothiazines and hydro-derivatives.
    상세보기
  7. Horwell David Christopher,GBX ; Bryans Justin S.,GBX ; Kneen Clare O.,GBX ; Morrell Andrew I.,GBX ; Ratcliffe Giles S.,GBX, Bridged cyclic amino acids as pharmaceutical agents.
    상세보기
  8. Khanna Satish C. (Bottmingen CHX), Coated adhesive tablets.
    상세보기
  9. Rice Ken Duane ; Dener Jeffrey Mark ; Gangloff Anthony Robert ; Kuo Elaine Yee-Lin, Compositions and methods for treating mast-cell mediated conditions.
    상세보기
  10. Mehta Atul M. (252 E. Crescent Ave. Ramsey NJ 07446), Controlled release indomethacin.
    상세보기
  11. Yatvin Milton B. ; Stowell Michael H. B. ; Meredith Michael J., Covalent polar lipid conjugates with neurologically active compounds for targeting.
    상세보기
  12. Sinnreich Joel (Basel CHX), Covered retard forms.
    상세보기
  13. Satzinger Gerhard (Denzlingen DT) Hartenstein Johannes (Wittental DT) Herrmann Manfred (St. Peter DT) Heldt Wolfgang (Wasser DT), Cyclic amino acids.
    상세보기
  14. Borchardt Ronald T. (Lawrence KS) Siahaan Teruna (Lawrence KS) Gangwar Sanjeev (Lawrence KS) Stella Valentino J. (Lawrence KS) Wang Binghe (Norman OK), Cyclic prodrugs of peptides and peptide nucleic acids having improved metabolic stability and cell membrane permeability.
    상세보기
  15. Urquhart John (Palo Alto CA) Theeuwes Felix (Los Altos CA), Delivery system comprising means for shielding a multiplicity of reservoirs in selected environment of use.
    상세보기
  16. Myers, Robert F., Derivatives of ampicillin and amoxicillin with beta-lactamase inhibitors.
    상세보기
  17. Alexander Jose (Lawrence KS), Dioxolenylmethyl carbamates pro moieties for amine drugs.
    상세보기
  18. Ayer Atul D. (Palo Alto CA) Swanson David R. (Palo Alto CA) Kuczynski Anthony L. (Palo Alto CA), Dosage form for treating cardiovascular diseases comprising isradipine.
    상세보기
  19. Choi ; Nam Sok ; Heller ; Jorge, Drug delivery devices manufactured from poly(orthoesters) and poly(orthocarbonates).
    상세보기
  20. Urquhart John (Palo Alto CA) Theeuwes Felix (Los Altos CA), Drug delivery system comprising a reservoir containing a plurality of tiny pills.
    상세보기
  21. Bodor Nicholas S. (Lawrence KS) Zupan Jack A. (Lawrence KS), Esters of cromoglycates.
    상세보기
  22. Duggan Mark E. (Schwenksville PA) Egbertson Melissa S. (Ambler PA) Ihle Nathan (Perkasie PA) Hartman George D. (Lansdale PA) Turchi Laura M. (Broomall PA) Hoffman William F. (Lansdale PA), Fibrinogen receptor antagonists for inhibiting aggregation of blood platelets.
    상세보기
  23. Bueno Lionel,FRX ; Chovet Maria,FRX ; Diop Laurent,FRX ; Guglietta Antonio ; Little Hilary J.,GBX ; Rafferty Michael Francis ; Ren Jiayuan ; Taylor ; Jr. Charles Price ; Watson William P.,GBX, GABA analogs to prevent and treat gastrointestinal damage.
    상세보기
  24. Silverman Richard B. (Morton Grove IL) Andruszkiewicz Ryszard (Sopot PLX) Yuen Po-Wai (Ann Arbor MI) Sobieray Denis M. (Holland MI) Franklin Lloyd C. (Hamilton MI) Schwindt Mark A. (Holland MI), GABA and L-glutamic acid analogs for antiseizure treatment.
    상세보기
  25. Silverman Richard B. (Morton Grove IL) Andruszkiewicz Ryszard (Sopot PLX) Yuen Po-Wai (Ann Arbor MI) Sobieray Denis M. (Holland MI) Franklin Lloyd C. (Hamilton MI) Schwindt Mark A. (Holland MI), GABA and L-glutamic acid analogs for antiseizure treatment.
    상세보기
  26. Silverman Richard B. ; Andruszkiewicz Ryszard,PLX ; Yuen Po-Wai ; Sobieray Denis Martin ; Franklin Lloyd Charles ; Schwindt Mark Alan, GABA and L-glutamic acid analogs for antiseizure treatment.
    상세보기
  27. Silverman Richard B. ; Andruszkiewicz Ryszard,PLX ; Yuen Po-Wai ; Sobieray Denis Martin ; Franklin Lloyd Charles ; Schwindt Mark Alan, GABA and L-glutamic acid analogs for antiseizure treatment.
    상세보기
  28. Shashoua Victor E. (Brookline MA), GABA esters and GABA analog esters.
    상세보기
  29. Singh Lakhbir,GBX, Isobutylgaba and its derivatives for the treatment of pain.
    상세보기
  30. Augart Helmut,DEX ; Gebhardt Uwe,DEX ; Herrmann Wolfgang,DEX, Lactam-free amino acids.
    상세보기
  31. Ferres Harry (Horsham EN) Clayton John Peter (Horsham EN), Lactonyl esters of penicillins.
    상세보기
  32. Theeuwes Felix (Los Altos CA), Method for adminstering tiny pills.
    상세보기
  33. Chien Yie W. (Skokie IL) Lambert Howard J. (Deerfield IL), Method for making a microsealed delivery device.
    상세보기
  34. Grosswald Ralph R. (Fairfield IA) Anderson Jeffory B. (Springville UT) Andrew Clair S. (Provo UT), Method for the manufacture of pharmaceutical cellulose capsules.
    상세보기
  35. Benedikt ; Gerald, New oral form of medicament and a method for producing it.
    상세보기
  36. Woodruff Geoffrey N. (Herts GBX), Novel methods for treating neurodegenerative diseases.
    상세보기
  37. Ayer Atul D. (Mountain View CA) Theeuwes Felix (Los Altos CA), Osmotic system with distribution zone for dispensing beneficial agent.
    상세보기
  38. Shtohryn Liudoslava V. (Budd Lake NJ) Peters David (Long Valley NJ), Pharmaceutical composition.
    상세보기
  39. Choi ; Nam Sok ; Heller ; Jorge, Poly(carbonates).
    상세보기
  40. Schmitt ; Edward Emil, Poly(orthoester) co- and homopolymers and poly(orthocarbonate) co- and homopolymers having carbonyloxy functionality.
    상세보기
  41. Capozza ; Richard C., Polymeric orthoesters housing beneficial drug for controlled release therefrom.
    상세보기
  42. Theeuwes ; Felix ; Saunders ; Richard J. ; Mefford ; Wayne S., Process for forming outlet passageways in pills using a laser.
    상세보기
  43. Ayer Atul D. (Mountain View CA) Theeuwes Felix (Los Altos CA), Process for manufacturing device with dispersion zone.
    상세보기
  44. Joseph Joachim FR; Pascal Prindirre FR; Nabil Farah FR, Process for manufacturing tablets for the sustained release of active principle(s).
    상세보기
  45. Alexander Jose (Lawrence KS), Process for preparing novel N-(acyloxy-alkoxy)carbonyl derivatives useful as bioreversible prodrug moieties for primary.
    상세보기
  46. Nabil Farah FR; Philippe Barthelemy FR; Joseph Joachim FR, Process for the manufacture of pharmaceutical composition with modified release of active principle comprising the matrix.
    상세보기
  47. Chu Daniel T. (Santa Clara CA) Li Qun (Gurnee IL) Cooper Curt S. (Gurnee IL) Fung Anthony K. L. (Gurnee IL) Lee Cheuk M. (Libertyville IL) Plattner Jacob J. (Libertyville IL), Quinolizinone type compounds.
    상세보기
  48. Michaels Alan S. (Atherton CA), Structured bioerodible drug delivery device.
    상세보기
  49. Horwell David Christopher,GBX ; Bryans Justin S.,GBX ; Kneen Clare O.,GBX ; Morrell Andrew I.,GBX ; Ratcliffe Giles S.,GBX ; Hartenstein Johannes,DEX, Substituted cyclic amino acids as pharmaceutical agents.
    상세보기
  50. Walters Eugene L. (Cincinnati OH), Sustained release diethylpropion compositions.
    상세보기
  51. Roussin Pascale,FRX ; Duddu Sarma, Sustained release theophylline formulations, excipient systems and methods of production.
    상세보기
  52. Hale Ron L. (Woodside CA) Lu Amy T. (Los Altos CA) Solas Dennis W. (San Francisco CA) Cormier Michel J. N. (Mountain View CA), Testosterone prodrugs for improved drug delivery.
    상세보기
  53. Satzinger ; Gerhard ; Hartenstein ; Johannes ; Herrmann ; Manfred ; Hel dt ; Wolfgang, Treatment of cranial dysfunctions using novel cyclic amino acids.
    상세보기
  54. Biesalski Hans K. (Albig DEX), Vitamin A aerosol-inhalant preparations and method.
    상세보기
  55. Biesalski Hans K. (Albig DEX), Vitamin A aerosol-inhalate preparations.
    상세보기

이 특허를 인용한 특허 (23)

  1. Dai, Xuedong; Gangakhedkar, Archana; Xiang, Jia Ning; Gallop, Mark A, Acyloxyalkyl carbamate prodrugs of α-amino acids, methods of synthesis and use.
    상세보기
  2. Dai, Xuedong; Gangakhedkar, Archana; Xiang, Jia-Ning; Gallop, Mark A, Acyloxyalkyl carbamate prodrugs of α-amino acids, methods of synthesis and use.
    상세보기
  3. Gallop, Mark A.; Yao, Fenmei; Ludwikow, Maria J.; Phan, Thu; Peng, Ge, Acyloxyalkyl carbamate prodrugs, methods of synthesis and use.
    상세보기
  4. Yao, Fenmei; Gallop, Mark A.; Barrett, Ronald W.; Virsik, Peter A., Crystalline form of a (3S)-aminomethyl-5-methyl-hexanoic acid prodrug and methods of use.
    상세보기
  5. Yao, Fenmei; Gallop, Mark A.; Barrett, Ronald W.; Virsik, Peter A., Crystalline form of a (3S)-aminomethyl-5-methyl-hexanoic acid prodrug and methods of use.
    상세보기
  6. Estrada, Tono; Raillard, Stephen P., Crystalline form of γ-aminobutyric acid analog.
    상세보기
  7. Estrada, Tono; Raillard, Stephen P.; Frauenfelder, Christine; Zacher, Uwe, Crystalline form of γ-aminobutyric acid analog.
    상세보기
  8. Estrada, Tono; Raillard, Stephen P.; Frauenfelder, Christine; Zacher, Uwe, Crystalline form of γ-aminobutyric acid analog.
    상세보기
  9. Gallop, Mark A.; Yao, Fenmei; Ludwikow, Maria J.; Peng, Ge; Raillard, Stephen P., Enantiomerically resolving acyloxyalkyl thiocarbonates used in synthesizing acyloxyalkyl carbamate prodrugs.
    상세보기
  10. Cundy, Kenneth C.; Sastry, Srikonda; Leung, Manshiu; Kadri, Balaji V.; Stach, Paul E., GABA analog prodrug sustained release oral dosage forms.
    상세보기
  11. Yao, Fenmei; Gallop, Mark A.; Barrett, Ronald W.; Virsik, Peter A., Mesophasic forms of (3S)-aminomethyl-5-methyl-hexanoic acid prodrugs and methods of use.
    상세보기
  12. Bhat, Laxminarayan; Gallop, Mark A., Methods for synthesis of acyloxyalkyl compounds.
    상세보기
  13. Bhat, Laxminarayan; Gallop, Mark A., Methods for synthesis of acyloxyalkyl compounds.
    상세보기
  14. Raillard, Stephen P.; Manthati, Suresh K.; Liu, Peng; Dai, Qunying; Yin, Hao, Methods of synthesizing .
    상세보기
  15. Raillard, Stephen P.; Manthati, Suresh K.; Liu, Peng; Dai, Qunying; Yin, Hao, Methods of synthesizing 1-(acyloxy)-alkyl carbamate prodrugs.
    상세보기
  16. Gallop, Mark A.; Cundy, Kenneth C.; Zhou, Cindy X.; Yao, Fenmei; Xiang, Jia-Ning, Methods of using prodrugs of pregabalin.
    상세보기
  17. Ben Moha-Lerman, Elena; Nidam, Tamar; Cohen, Meital; Avhar-Maydan, Sharon; Balanov, Anna, Processes for the preparation and purification of gabapentin enacarbil.
    상세보기
  18. Gallop, Mark A.; Cundy, Kenneth C.; Zhou, Cindy X.; Qiu, Fayang G.; Yao, Fenmei; Xiang, Jia-Ning; Ollmann, Ian R., Prodrugs of GABA analogs, compositions and uses thereof.
    상세보기
  19. Gallop, Mark A.; Cundy, Kenneth C.; Zhou, Cindy X.; Yao, Fenmei; Xiang, Jia-Ning, Prodrugs of GABA analogs, compositions and uses thereof.
    상세보기
  20. Gallop, Mark A.; Cundy, Kenneth C.; Zhou, Cindy X.; Yao, Fenmei; Xiang, Jia-Ning; Ollman, Ian R.; Qiu, Fayang G., Prodrugs of GABA analogs, compositions and uses thereof.
    상세보기
  21. Gallop, Mark A., Prodrugs of gaba analogs, compositions and uses thereof.
    상세보기
  22. Edgren, David E.; Kidney, David J.; Pargaonkar, Nikhil; Kim, Derrick K.; Yoder, Gorm; Karaborni, Sarni, Sustained release oral dosage forms of an R-baclofen prodrug.
    상세보기
  23. Barrett, Ronald W., Treating urinary incontinence using prodrugs of GABA analogs.
    상세보기

관련 콘텐츠

섹션별 컨텐츠 바로가기

AI-Helper ※ AI-Helper는 오픈소스 모델을 사용합니다.

AI-Helper 아이콘
AI-Helper
안녕하세요, AI-Helper입니다. 좌측 "선택된 텍스트"에서 텍스트를 선택하여 요약, 번역, 용어설명을 실행하세요.
※ AI-Helper는 부적절한 답변을 할 수 있습니다.

선택된 텍스트

맨위로