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Medicaments comprising betamimetics and a novel anticholinergic 원문보기

IPC분류정보
국가/구분 United States(US) Patent 등록
국제특허분류(IPC7판)
  • A61K-009/08
  • A61K-009/10
  • A61K-009/12
  • A61K-009/14
  • A61K-009/48
  • A61K-031/40
  • A61K-031/336
  • A61K-031/438
  • A61K-031/439
  • C07D-451/00
  • C07D-451/02
출원번호 US-0395501 (2003-03-24)
등록번호 US-7417051 (2008-08-26)
우선권정보 DE-102 16 428(2002-04-12); DE-102 56 317(2002-12-03)
발명자 / 주소
  • Banholzer,Rolf
  • Meissner,Helmut
  • Morschhaeuser,Gerd
  • Pieper,Michael P.
  • Pohl,Gerald
  • Reichl,Richard
  • Speck,Georg
  • Meade,Christopher John Montague
  • Pairet,Michel
  • Konetzki,Ingo
출원인 / 주소
  • Boehringer Ingelheim Pharma GmbH & Co. KG
대리인 / 주소
    Morris,Michael P.
인용정보 피인용 횟수 : 24  인용 특허 : 11

초록

A pharmaceutical composition comprising: (a) a salt of formula 1 wherein: X- is an anion with a single negative charge; and (b) a betamimetic 2, or a solvate or hydrate thereof, optionally in the form of the enantiomers, mixtures of the enantiomers, or in the form of the racemates thereof, p

대표청구항

We claim: 1. A pharmaceutical composition comprising: (a) a salt of formula 1 wherein: X- is an anion with a single negative charge; and (b) a betamimetic 2 wherein the betamimetic 2 is a salmeterol salt, formoterol salt, or acid addition salt of a compound of formula 2a' wherein: R1 and R2

이 특허에 인용된 특허 (11)

  1. Meissner, Helmut; Morschhaeuser, Gerd; Pieper, Michael Paul; Pohl, Gerald; Reichl, Richard; Speck, Georg; Banholzer, Rolf, Anticholinergics which may be used as medicaments as well as processes for preparing them.
  2. Banholzer Rolf,DEX ; Bauer Rudolf,DEX ; Reichl Richard,DEX, Esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions.
  3. Banholzer Rolf (Ingelheim am Rhein DEX) Bauer Rudolf (Ockenheim DEX) Reichl Richard (Gau-Algesheim DEX), Esters of bi-and tricyclic amino alcohols and their use in pharmaceutical compositions.
  4. Banholzer Rolf (Ingelheim am Rheim DEX) Bauer Rudolf (Wiesbaden DEX) Reichl Richard (Ingelheim am Rheim DEX), Esters of thienyl carboxylic acids and amino alcohols and their quaternization products.
  5. Banholzer Rolf (Ingelheim am Rhein DEX), N-alkylnorscopines and acid addition salts thereof.
  6. Banholzer, Rolf; Graulich, Manfred; Luettke, Sven; Mathes, Andreas; Meissner, Helmut; Specht, Peter; Broeder, Wolfgang, Process for preparing a scopine ester intermediate.
  7. Rolf Banholzer DE; Manfred Graulich DE; Sven Luettke DE; Andreas Mathes DE; Helmut Meissner DE; Peter Specht DE; Wolfgang Broeder DE, Process for preparing an anticholinergic.
  8. Banholzer Rolf,DEX, Process for preparing pure enantiomers of tropic acid esters.
  9. Brandenburg, Joerg; Pfrengle, Waldemar Franz-Augustin; Rall, Werner, Process for preparing scopine esters.
  10. Banholzer Rolf (Ingelheim DEX) Bauer Rudolf (Wiesbaden DEX), Quaternary 6,11-dihydro-dibenzo-[b,e]-thiepine-11-N-alkylnorscopine ethers having spasmolytic activity.
  11. Banholzer Rolf (Ingelheim am Rhein DT) Bauer Rudolf (Wiesbaden DT) Heusner Alex (Gau-Algesheim DT) Schulz Werner (Ingelheim am Rhein DT), Quaternary N-b 상세보기

이 특허를 인용한 특허 (24)

  1. Wachtel, Herbert, Adapter, inhalation device, and atomizer.
  2. Eicher, Joachim; Graessl, Herbert; Janetzko, Mike; Jung, Andree; Meisenheimer, Martin; Wachtel, Herbert; Winkler, Robert Gerhard; Wuttke, Gilbert; Yu, Ying, Container, nebulizer and use.
  3. Besseler, Jens; Holakovsky, Holger; Argauer, Herbert; Gatz, Josef; Gorshoefer, Andreas, Dispenser with encoding means.
  4. Dunne, Stephen T.; Moser, Achim, Dispensing device, storage device and method for dispensing a formulation.
  5. Lustenberger, Philipp; Konetzki, Ingo; Sieger, Peter, Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments.
  6. Bhide, Vishwajit; Amperayani Pattabhi, Raghuram; Pimple, Rohini; Choubey, Bishu, Inhaler.
  7. Bhide, Vishwajit; Amperayani Pattabhi, Raghuram; Pimple, Rohini; Choubey, Bishu, Inhaler.
  8. Grauert, Matthias; Bouyssou, Thierry; Lustenberger, Philipp; Breitfelder, Steffen; Schnapp, Andreas; Pieper, Michael P.; Rudolf, Klaus; Speck, Georg, Long acting bronchodilators for the treatment of respiratory diseases.
  9. Konetzki, Ingo; Schromm, Kurt; Schollenberger, Hermann; Pestel, Sabine; Schnapp, Andreas; Bouyssou, Thierry; Buettner, Frank; Heine, Claudia; Lustenberger, Philipp; Hoenke, Christoph; Rudolf, Klaus, Medicaments for the treatment of chronic obstructive pulmonary disease.
  10. Konetzki, Ingo; Schromm, Kurt; Schollenberger, Hermann; Pestel, Sabine; Schnapp, Andreas; Bouyssou, Thierry; Buettner, Frank; Heine, Claudia; Lustenberger, Philipp; Hoenke, Christoph; Rudolf, Klaus, Medicaments for the treatment of chronic obstructive pulmonary disease.
  11. Konetzki, Ingo; Schromm, Kurt; Schollenberger, Hermann; Pestel, Sabine; Schnapp, Andreas; Bouyssou, Thierry; Buettner, Frank; Heine, Claudia; Rudolf, Klaus; Lustenberger, Philipp; Hoenke, Christoph, Medicaments for the treatment of chronic obstructive pulmonary disease.
  12. Holakovsky, Holger; Lange, Lars; Steinzen, Maurice; Weiland, Felix; List, Klaus, Medicinal device with container.
  13. Schuy, Steffen; Meisenheimer, Martin; Witte, Florian, Method for coating a surface of a component.
  14. Besseler, Jens; Holakovsky, Holger; Gorshoefer, Andreas; Gatz, Josef; Argauer, Herbert, Nebuliser with coding means.
  15. Bach, Alexander; Besseler, Jens; Holakovsky, Holger; Daelman, Manuel; Wuttke, Gilbert, Nebulizer.
  16. Bach, Alexander; Besseler, Jens; Holakovsky, Holger; Daelman, Manuel; Wuttke, Gilbert; Frenkel, Udo, Nebulizer.
  17. Bach, Alexander; Besseler, Jens; Holakovsky, Holger; Kaemper, Markus; Krakowka, Manuel; Wuttke, Gilbert, Nebulizer.
  18. Besseler, Jens; Herrmann, Frank; Holakovsky, Holger; Argauer, Herbert; Gatz, Josef; Gorshoefer, Andreas, Nebulizer.
  19. Besseler, Jens; Herrmann, Frank; Holakovsky, Holger; Argauer, Herbert; Gatz, Josef; Gorshoefer, Andreas, Nebulizer.
  20. Eicher, Joachim; Gatz, Josef; Herrmann, Frank; Hoelz, Hubert; Jung, Andree; Meisenheimer, Martin; Mueller, Markus; Von Schuckmann, Alfred; Wachtel, Herbert; Winkler, Robert Gerhard; Wuttke, Gilbert; Ziegler, Jochen, Nebulizer.
  21. Herrmann, Frank; Krenz, Holger; Endert, Guido; Wergen, Horst, Nebulizer.
  22. Holakovsky, Holger; Thoemmes, Ralf; Rohrschneider, Marc; Witte, Florian; Deane, Kevin Peter; Jennings, Douglas Ivan, Nebulizer.
  23. Krueger, Thomas; Ries, Uwe; Schnaubelt, Juergen; Rall, Werner; Leuter, Zeno A.; Duran, Adil; Soyka, Rainer, Process for the manufacturing of betamimetics.
  24. Fairhurst, Robin Alec; Sandham, David Andrew; Beattie, David; Bruce, Ian; Cuenoud, Bernard; Madden, Reamonn; Press, Neil John; Taylor, Roger John; Turner, Katharine Louise; Watson, Simon James, Quinoline-2-one derivatives for the treatment of airways diseases.
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