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NTIS 바로가기Bulletin of the Korean chemical society, v.30 no.6, 2009년, pp.1313 - 1316
Park, Hwang-Seo (Department of Bioscience and Biotechnology, Sejong University) , Jung, Suk-Kyeong (Medical Proteomics Research Center, Korea Research Institute of Bioscience and Biotechnology) , Bahn, Young-Jae (Medical Proteomics Research Center, Korea Research Institute of Bioscience and Biotechnology) , Jeong, Dae-Gwin (Medical Proteomics Research Center, Korea Research Institute of Bioscience and Biotechnology) , Ryu, Seong-Eon (Department of Bio-engineering, Hanyang University) , Kim, Seung-Jun (Medical Proteomics Research Center, Korea Research Institute of Bioscience and Biotechnology)
Cdc25 phosphatases have been considered as attractive drug targets for anticancer therapy due to the correlation of their overexpression with a wide variety of cancers. We have been able to identify five novel Cdc25 phosphatase inhibitors with micromolar activity by means of a structure-based de nov...
Kristjansdottir, K.; Rudolph, J. Chem. Biol. 2004, 11, 1043.
Rudolph, J. Biochemistry 2007, 46, 3595.
Galaktionov, K.; Lee, A. K.; Eckstein, J.; Draetta, G.; Meckler, J.; Loda, M.; Beach, D. Science 1995, 269, 1575.
Takemara, I.; Yamamoto, H.; Sekimoto, M.; Ohue, M.; Noura, S.; Miyake, Y.; Matsumoto, T.; Aihara, T.; Tomita, N.; Tamaki, Y.; Sakita, I.; Kikkawa, N.; Matsuura, N.; Shiozaki, H.; Monden, M. Cancer Res. 2000, 60, 3043.
Ngan, E. S. W.; Hashimoto, Y.; Ma, Z.-Q.; Tsai, M. J.; Tsai, S. Y. Oncogene 2003, 22, 734.
Boutros, R.; Dozier, C.; Ducommun, B. Curr. Opin. Cell Biol. 2006, 18, 185.
Fauman, E. B.; Cogswell, J. P.; Lovejoy, B.; Rocque, W. J.; Holmes, W.; Montana, V. G.; Piwnica-Worms, H.; Rink, M. J.; Saper, M. A. Cell 1998, 93, 617.
Reynolds, R. A.; Yem, A. W.; Wolfe, C. L.; Deibel, M. R.; Chidester, C. G.; Watenpaugh, K. D. J. Mol. Biol. 1999, 293, 559.
Contour-Galcera, M.-O.; Sidhu, A.; Prevost, G.; Bigg, D.; Ducommun, B. Pharmcol. Ther. 2007, 115, 1.
Ham, S. W.; Carr, B. I. Drug Des. Rev. 2004, 1, 123.
Lazo, J. S.; Aslan, D. C.; Southwick, E. C.; Cooley, K. A.; Ducruet, A. P.; Joo, B.; Vogt, A.; Wipf, P. J. Med. Chem. 2001, 44, 4042.
Sohn, J.; Kiburz, B.; Li, Z.; Deng, L.; Safi, A.; Pirrung, M. C.; Rudolph, J. J. Med. Chem. 2003, 46, 2580.
Brault, L.; Denance, M.; Banaszak, E.; Maadidi, S. E.; Battaglia, E.; Bagrel, D.; Samadi, M. Eur. J. Med. Chem. 2007, 42, 243.
Huang, W.; Li, J.; Zhang, W.; Zhou, Y.; Xie, C.; Luo, Y.; Li, Y.; Wang, J.; Li, J.; Lu, W. Bioorg. Med. Chem. Lett. 2006, 16, 1905.
Lazo, J. S.; Nemoto, K.; Pestell, K. E.; Cooley, K.; Southwick, E. C.; Mitchell, D. A.; Furey, W.; Gussio, R.; Zaharevitz, D.W.; Joo, B.; Wipf, P. Mol. Pharmacol. 2002, 61, 720.
Lavecchia, A.; Cosconati, S.; Limongelli, V.; Novellino, E. Chem. Med. Chem 2006, 1, 540.
Park, H.; Carr, B. I.; Li, M.; Ham, S. W. Bioorg. Med. Chem. Lett. 2007, 17, 2351.
Park, H.; Bahn, Y. J.; Jung, S.-K.; Jeong, D. G.; Lee, S.-H.; Seo, I.; Yoon, T.-S.; Kim, S. J.; Ryu, S. E. J. Med. Chem. 2008, 51, 5533.
Shoichet, B. K.; Leach, A. R.; Kuntz, I. D. Proteins 1999, 34, 4.
Wang, R.; Gao, Y.; Lai, L. J. Mol. Model. 2000, 6, 498.
Wang, R.; Liu, L.; Lai, L. J. Mol. Model. 1998, 6, 379.
Gasteiger, J.; Marsili, M. Tetrahedron 1980, 36, 3219.
Kang, H.; Choi, H.; Park, H. J. Chem. Inf. Model. 2007, 47, 509.
Morris, G. M.; Goodsell, D. S.; Halliday, R. S.; Huey, R.; Hart, W. E.; Belew, R. K.; Olson, A. J. J. Comput. Chem. 1998, 19, 1639.
Lipinski, C. A.; Lombardo, F.; Dominy, B. W.; Feeney, P. J. Adv. Drug. Delivery. Rev. 1997, 23, 3.
Tamura, K.; Southwick, E. C.; Kerns, J.; Rosi, K.; Carr, B. I.; Wilcox, C.; Lazo, J. S. Cancer Res. 2000 60, 1317.
Osada, S.; Osada, K.; Carr, B. I. J. Mol. Biol. 2001, 314, 765.
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